BF3·OEt2-catalyzed one-pot three-component access to diarylmethylazides

Sure Siva Prasad; Dirgha Raj Joshi; Ikyon Kim

doi:10.1016/j.tetlet.2020.152820

BF₃·OEt₂-catalyzed one-pot three-component access to diarylmethylazides

Sure Siva Prasad, Dirgha Raj Joshi, Ikyon Kim

Department of Pharmacy

Research output: Contribution to journal › Article › peer-review

Abstract

A direct one-pot access to diarylmethylazides, versatile intermediates, from commercially available starting materials was enabled via three-component coupling of aldehydes, arenes, and TMSN₃ in the presence of a catalytic amount of BF₃·OEt₂.

Original language	English
Article number	152820
Journal	Tetrahedron Letters
Volume	67
DOIs	https://doi.org/10.1016/j.tetlet.2020.152820
Publication status	Published - 2021 Mar 16

Bibliographical note

Funding Information:
We thank the National Research Foundation of Korea ( NRF-2018R1A6A1A03023718 and NRF-2020R1A2C2005961 ) for generous financial support.

Publisher Copyright:
© 2021 Elsevier Ltd

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

Access to Document

10.1016/j.tetlet.2020.152820

Cite this

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title = "BF3·OEt2-catalyzed one-pot three-component access to diarylmethylazides",

abstract = "A direct one-pot access to diarylmethylazides, versatile intermediates, from commercially available starting materials was enabled via three-component coupling of aldehydes, arenes, and TMSN3 in the presence of a catalytic amount of BF3·OEt2.",

author = "Prasad, {Sure Siva} and Joshi, {Dirgha Raj} and Ikyon Kim",

note = "Funding Information: We thank the National Research Foundation of Korea ( NRF-2018R1A6A1A03023718 and NRF-2020R1A2C2005961 ) for generous financial support. Publisher Copyright: {\textcopyright} 2021 Elsevier Ltd",

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