Facile approach to diverse 3-acylated indolizines via a sequential Sonogashira coupling/iodocyclization process

Youngeun Jung, Ikyon Kim

Research output: Contribution to journalArticle

19 Citations (Scopus)

Abstract

Successful implementation of a sequential Pd-catalyzed Sonogashira cross-coupling/iodine-promoted 5-exo-dig cyclization procedure with pyridines bearing a terminal alkyne moiety provided direct and straightforward access to a diverse array of 3-acylated indolizines under mild conditions.

Original languageEnglish
Pages (from-to)8198-8206
Number of pages9
JournalTetrahedron
Volume68
Issue number39
DOIs
Publication statusPublished - 2012 Sep 30

Fingerprint

Indolizines
Bearings (structural)
Pyridines
Alkynes
Cyclization
Iodine

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry

Cite this

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Facile approach to diverse 3-acylated indolizines via a sequential Sonogashira coupling/iodocyclization process. / Jung, Youngeun; Kim, Ikyon.

In: Tetrahedron, Vol. 68, No. 39, 30.09.2012, p. 8198-8206.

Research output: Contribution to journalArticle

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