Highly selective catalytic Friedel-Crafts acylation and sulfonylation of activated aromatic compounds using indium metal

Doo Ok Jang; Kyung Soo Moon; Dae Hyan Cho; Joong Gon Kim

doi:10.1016/j.tetlet.2006.06.099

Highly selective catalytic Friedel-Crafts acylation and sulfonylation of activated aromatic compounds using indium metal

Doo Ok Jang, Kyung Soo Moon, Dae Hyan Cho, Joong Gon Kim

Chemistry and Medical Chemistry

Research output: Contribution to journal › Article › peer-review

52 Citations (Scopus)

Abstract

The Friedel-Crafts acylation of activated benzenes with various aromatic and aliphatic acid chlorides was studied in the presence of indium metal. The reaction was accomplished in high isolated yields under solvent or solvent-less conditions. The method is also applicable for preparing diaryl sulfones from aromatic compounds and aryl sulfonyl chlorides.

Original language	English
Pages (from-to)	6063-6066
Number of pages	4
Journal	Tetrahedron Letters
Volume	47
Issue number	34
DOIs	https://doi.org/10.1016/j.tetlet.2006.06.099
Publication status	Published - 2006 Aug 21

Bibliographical note

Funding Information:
This work was supported by the Center for Bioactive Molecular Hybrids and Yonsei University.

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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title = "Highly selective catalytic Friedel-Crafts acylation and sulfonylation of activated aromatic compounds using indium metal",

abstract = "The Friedel-Crafts acylation of activated benzenes with various aromatic and aliphatic acid chlorides was studied in the presence of indium metal. The reaction was accomplished in high isolated yields under solvent or solvent-less conditions. The method is also applicable for preparing diaryl sulfones from aromatic compounds and aryl sulfonyl chlorides.",

author = "Jang, {Doo Ok} and Moon, {Kyung Soo} and Cho, {Dae Hyan} and Kim, {Joong Gon}",

note = "Funding Information: This work was supported by the Center for Bioactive Molecular Hybrids and Yonsei University.",

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T1 - Highly selective catalytic Friedel-Crafts acylation and sulfonylation of activated aromatic compounds using indium metal

AU - Jang, Doo Ok

AU - Moon, Kyung Soo

AU - Cho, Dae Hyan

AU - Kim, Joong Gon

N1 - Funding Information: This work was supported by the Center for Bioactive Molecular Hybrids and Yonsei University.

PY - 2006/8/21

Y1 - 2006/8/21

N2 - The Friedel-Crafts acylation of activated benzenes with various aromatic and aliphatic acid chlorides was studied in the presence of indium metal. The reaction was accomplished in high isolated yields under solvent or solvent-less conditions. The method is also applicable for preparing diaryl sulfones from aromatic compounds and aryl sulfonyl chlorides.

AB - The Friedel-Crafts acylation of activated benzenes with various aromatic and aliphatic acid chlorides was studied in the presence of indium metal. The reaction was accomplished in high isolated yields under solvent or solvent-less conditions. The method is also applicable for preparing diaryl sulfones from aromatic compounds and aryl sulfonyl chlorides.

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U2 - 10.1016/j.tetlet.2006.06.099

DO - 10.1016/j.tetlet.2006.06.099

M3 - Article

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VL - 47

SP - 6063

EP - 6066

JO - Tetrahedron Letters

JF - Tetrahedron Letters

SN - 0040-4039

IS - 34

ER -

Highly selective catalytic Friedel-Crafts acylation and sulfonylation of activated aromatic compounds using indium metal

Abstract

Bibliographical note

All Science Journal Classification (ASJC) codes

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