Indium-mediated mild and facile method for the synthesis of amides

Dae Hyan Cho; Doo Ok Jang

doi:10.1016/j.tetlet.2004.01.114

Indium-mediated mild and facile method for the synthesis of amides

Dae Hyan Cho, Doo Ok Jang

Chemistry and Medical Chemistry

Research output: Contribution to journal › Article › peer-review

27 Citations (Scopus)

Abstract

Indium-mediated coupling reactions of acyl chlorides and amines for the synthesis of amide bonds are described. The reaction afforded high yields of the desired amides under mild and neutral conditions, and it was applicable also to the preparation of peptides without epimerization.

Original language	English
Pages (from-to)	2285-2287
Number of pages	3
Journal	Tetrahedron Letters
Volume	45
Issue number	11
DOIs	https://doi.org/10.1016/j.tetlet.2004.01.114
Publication status	Published - 2004 Feb 8

Bibliographical note

Funding Information:
This work was supported by Center for Bioactive Molecular Hybrids at Yonsei University.

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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title = "Indium-mediated mild and facile method for the synthesis of amides",

abstract = "Indium-mediated coupling reactions of acyl chlorides and amines for the synthesis of amide bonds are described. The reaction afforded high yields of the desired amides under mild and neutral conditions, and it was applicable also to the preparation of peptides without epimerization.",

author = "Cho, {Dae Hyan} and Jang, {Doo Ok}",

note = "Funding Information: This work was supported by Center for Bioactive Molecular Hybrids at Yonsei University.",

year = "2004",

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doi = "10.1016/j.tetlet.2004.01.114",

language = "English",

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AU - Cho, Dae Hyan

AU - Jang, Doo Ok

N1 - Funding Information: This work was supported by Center for Bioactive Molecular Hybrids at Yonsei University.

PY - 2004/2/8

Y1 - 2004/2/8

N2 - Indium-mediated coupling reactions of acyl chlorides and amines for the synthesis of amide bonds are described. The reaction afforded high yields of the desired amides under mild and neutral conditions, and it was applicable also to the preparation of peptides without epimerization.

AB - Indium-mediated coupling reactions of acyl chlorides and amines for the synthesis of amide bonds are described. The reaction afforded high yields of the desired amides under mild and neutral conditions, and it was applicable also to the preparation of peptides without epimerization.

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DO - 10.1016/j.tetlet.2004.01.114

M3 - Article

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VL - 45

SP - 2285

EP - 2287

JO - Tetrahedron Letters

JF - Tetrahedron Letters

SN - 0040-4039

IS - 11

ER -

Indium-mediated mild and facile method for the synthesis of amides

Abstract

Bibliographical note

All Science Journal Classification (ASJC) codes

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