Palladium-catalyzed α-arylation of aryloxyketones for the synthesis of 2,3-Disubstituted benzofurans

Jin Ho Lee, Myungock Kim, Ikyon Kim

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Abstract

A highly efficient palladium-catalyzed α-arylation of aryloxyketones has been developed, allowing for facile installation of various (hetero)aryl groups at C2 position in good to excellent yields. Subsequent cyclodehydration of the resulting α-arylated aryloxyketones provided rapid access to diverse 2,3-disubstitured benzofurans.

Original languageEnglish
Pages (from-to)6153-6163
Number of pages11
JournalJournal of Organic Chemistry
Volume79
Issue number13
DOIs
Publication statusPublished - 2014 Jul 3

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All Science Journal Classification (ASJC) codes

  • Organic Chemistry

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