Abstract
New glycosylated peptidomimetics possessing O- and N-glycosylated α-aminooxy acids were efficiently synthesized by fragment coupling on solid support. The N-terminal glycosylated tripeptide mimics prepared in solution were coupled to the C-terminal dipeptides attached to the resin under O-(7-azabenzotriazole-I-yl)-1, 1, 3, 3-tetramethyluronium hexafluorophosphate (HATU)/1-hydroxy-7-azabenzotriazole (HOAt)/N-ethylmorpholin (NEM) conditions.
| Original language | English |
|---|---|
| Pages (from-to) | 1463-1466 |
| Number of pages | 4 |
| Journal | Synlett |
| Issue number | 9 |
| DOIs | |
| Publication status | Published - 2002 |
All Science Journal Classification (ASJC) codes
- Organic Chemistry
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Lee, M. R., Lee, J., & Shin, I. (2002). Synthesis of novel glycopeptidomimetics containing O- and N-glycosylated α-aminooxy acids by fragment coupling on solid support. Synlett, (9), 1463-1466. https://doi.org/10.1055/s-2002-33509