TY - JOUR
T1 - Synthesis of novel glycopeptidomimetics containing O- and N-glycosylated α-aminooxy acids by fragment coupling on solid support
AU - Lee, Myung Ryul
AU - Lee, Jiyong
AU - Shin, Injae
N1 - Copyright:
Copyright 2018 Elsevier B.V., All rights reserved.
PY - 2002
Y1 - 2002
N2 - New glycosylated peptidomimetics possessing O- and N-glycosylated α-aminooxy acids were efficiently synthesized by fragment coupling on solid support. The N-terminal glycosylated tripeptide mimics prepared in solution were coupled to the C-terminal dipeptides attached to the resin under O-(7-azabenzotriazole-I-yl)-1, 1, 3, 3-tetramethyluronium hexafluorophosphate (HATU)/1-hydroxy-7-azabenzotriazole (HOAt)/N-ethylmorpholin (NEM) conditions.
AB - New glycosylated peptidomimetics possessing O- and N-glycosylated α-aminooxy acids were efficiently synthesized by fragment coupling on solid support. The N-terminal glycosylated tripeptide mimics prepared in solution were coupled to the C-terminal dipeptides attached to the resin under O-(7-azabenzotriazole-I-yl)-1, 1, 3, 3-tetramethyluronium hexafluorophosphate (HATU)/1-hydroxy-7-azabenzotriazole (HOAt)/N-ethylmorpholin (NEM) conditions.
UR - http://www.scopus.com/inward/record.url?scp=0036373849&partnerID=8YFLogxK
UR - http://www.scopus.com/inward/citedby.url?scp=0036373849&partnerID=8YFLogxK
U2 - 10.1055/s-2002-33509
DO - 10.1055/s-2002-33509
M3 - Article
AN - SCOPUS:0036373849
SP - 1463
EP - 1466
JO - Synlett
JF - Synlett
SN - 0936-5214
IS - 9
ER -